Imitsi Yongera Kurwanya Estrogene Steroide Ifu Yera Tamoxifen Citrate Nolvadex
Byihuse
Igicuruzwa: Nolvadex (Citrate ya Tamoxifen)
URUBANZA No: 54965-24-1
MF: C26H29NO
MW: 371.51
Isuku: 99%
Ingingo yo guteka: 482.3 ° C kuri 760 mmHg
Ububiko: Bifunze muri 2 ºC -8 ºC
Ingingo yo gushonga: 140-144 ° C.
flash point: 356.5ºC
Imiterere:
Einecs No: 234-118-0
Ibisanzwe: Ibipimo ngenderwaho
Ibindi bicuruzwa birwanya kanseri: Citrate ya Tamoxifen, Citrate ya Clomiphene, Citrate ya Toremifene, Anastrozole, Raloxifene hydrochloride, Fulvestrant, Letrozole, Crotamiton
Ikoreshwa: Tamoxifen ni imisemburo yumugore ishobora guhagarika ibikorwa bya estrogene, mubisanzwe ikoreshwa mukuvura ubwoko bumwe na bumwe bwa kanseri yamabere kubagabo nabagore.
Kuvura Kanseri Steroide dutanga
Citrate ya Tamoxifen | umukozi udafite steroidal |
Exemestane | inhibitor ya aromatase |
Anastrozole | ikoreshwa mugihe ukoresheje umubare munini wa aromatizing steroid |
Stanozolol | Gukata Amagare |
Toremifene Citrate | itari steroidal ihitamo Estrogen reseptor modulator |
Umuyoboro wa Drostanolone | Anabolic Steroid |
Methenolone Enanthate | protein hormone assimilation ibikorwa bikomeye byumwijima |
17-methyltestosterone | androgene na Albumen Assimilation steroid |
Fluoxymesterone | irashobora gukoreshwa nkibikoresho bya farumasi |
Formestan | Ikoreshwa nka aromatic enzyme inhibitor |
Nolvadex
Ifu: kuri garama 1 ya Citrate ya Tamoxifen
Umusaruro: Kwibanda cyane byakozwe - 20 mg / ml
Ibisabwa:
Garama 1 ya Citrate ya Tamoxifen
Inzoga 1 ikwiranye no gufata ingano yamazi
Miliyoni 19,6 za Glycerol
29.4 ml ya 190 Yerekana Inzoga
Ifu: kuri garama 1 ya Citrate ya Tamoxifen
Umusaruro: Kwibanda cyane byakozwe - 20 mg / ml
Ibisabwa:
Garama 1 ya Citrate ya Tamoxifen
Inzoga 1 ikwiranye no gufata ingano yamazi
9.8 ml ya PEG 600
39.2 ml ya 190 Yerekana Inzoga
Nolvadex Ikoreshwa na dosiye
Kanseri y'ibere | 10 mg 20 mg kumunwa kabiri kumunsi |
Kuri kanseri y'ibere | 20 mg 40 mg yatanzwe mugabanijwe |
Abagore bafite Carcinoma | 20 mg buri munsi kumyaka 5 |
Mugabanye kwandura kanseri y'ibere | 20mg buri munsi kumyaka 5 |
Kanseri y'ibere ya node nziza, gutandukana | 10 mg mu kanwa inshuro 2 kugeza kuri 3 kumunsi kumyaka 5. |
Abakobwa bafite imyaka 2 kugeza 10 hamwe na syndrome ya McCune-Albright | 20 mg buri munsi kumwaka umwe |
Porogaramu ya Nolvadex
1: Citrate ya Tamoxifen Koresha Kanseri
Tamoxifen citrate | Yemejwe gukumira: Kanseri y'ibere ku bagore bafite ibyago byinshi byo kurwara. |
Kanseri y'ibere ku bagore no ku bagabo | |
kwigwa mukuvura ubundi bwoko bwa kanseri. |
2: Inyungu za Tamoxifen
A. Tamoxifen itinda cyangwa ihagarika imikurire ya kanseri isanzwe igaragara mumubiri.Ifasha kurinda kanseri yumwimerere kutagaruka kandi ifasha kwirinda kanseri nshya mumabere atandukanye.Igabanya kandi ibyago byo kurwara kanseri y'ibere ku bagore bafite ibyago byinshi kuri iyi ndwara.
B. Tamoxifen ikoreshwa mukurinda no kuvura kanseri yamabere yipimisha neza kuri reseptor ya estrogene (ER +).Ihagarika ingaruka imisemburo ya estrogene igira kuri selile ya kanseri kandi igabanya amahirwe ya kanseri yamabere.Bikunze kwitwa "anti-estrogene."
C. Tamoxifen ifite akamaro kanini mukugabanya ibyago byo kongera kanseri y'ibere.Ku bagore bamaze kurwara kanseri y'ibere, tamoxifen nayo igabanya ibyago byo kurwara kanseri y'ibere mu ibere ritandukanye (impande zombi)
D. Kubagore nyuma yo gucura, kuvura ibyiciro bibiri ukoresheje tamoxifen hanyuma inhibitor ya aromatase, nka anastrozole (Arimidex), exemestane (Aromasin), cyangwa letrozole (Femara) irashobora gukora neza kuruta gufata tamoxifen gusa.