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ibicuruzwa

Igitsina gabo gisanzwe Steroid Hormone Igiti gikuramo Yohimbine Hcl Powder CAS 65-19-0

Ibisobanuro bigufi:


Ibisobanuro birambuye

Ibiranga ibicuruzwa

Byihuse

Izina ryibicuruzwa: Yohimbine HCl

Alias: Yohimbine Hydrochloride

URUBANZA OYA: 65-19-0

Einecs: 200-600-4

Isuku: 99%

Inzira ya molekulari: C21H27ClN2O

Uburemere bwa molekuline: 390.904

1

Kugaragara: Ifu yera ya kristaline, uburyohe bukaze.Irashobora gushonga muri chloroform, methanol, Ethanol, kandi igashonga gato mumazi.

Ikoreshwa:Yohimbineni imiti yimpuhwe na mydriaticKurikuvura ubudahangarwa ku barwayi b'igitsina gabo bafite inkomoko y'amaraso cyangwa diabete n'inkomoko ya psycogeneque.Yohimbineiraboneka munsi yamazina atandukanye akurikira: Aphrodyne, na Yocon.

Injiza Yohimbine Hcl

1g yo hcl.

1ml BA nka anesthetic, ariko nanone ikora bacstat.

9ml ya alcool.

90ml y'amazi yatoboye.

Reka gushonga muri BA na EA muminota 10 hanyuma wongeremo amazi bizagaragara ko ari ibicu nyuma yo kongeramo amazi, ariko ibyo ntacyo bitwaye kuko bizasa kimwe NYUMA anyuze mumashanyarazi ya 0.22.

Imikorere ya hydrohloride ya Yohimbine

(1).Kwihutisha ingufu z'umubiri metabolism no kongera ingufu;

(2).Kubyara imitekerereze ikangura ubushake bwo guhuza ibitsina;

(3).Kongera imitsi, hamwe numurimo wo guhagarika inkari nta nkomere.

Ibisobanuro

1. Hydrochloride ya Yohimbine yerekanwa nkimpuhwe na mydriatike.Irashobora kugira ibikorwa nka afrodisiac.

Ubudahangarwa (ntibushobora kugira erekisiyo)

Gukora mukongera umusaruro wumubiri wimiti ifasha kubyara.Ntabwo ikora mubagabo bose badafite imbaraga.

Ubushakashatsi bushya bwerekana ko bushobora kuba ibyatsi bifite imbaraga za antioxydeant.Ubushakashatsi bwerekana ko ari vasodilator, bivuze ko byongera umuvuduko wamaraso kuruhande no kumugereka.

2. Yohimbine byoroshye kwinjira muri (CNS) kandi itanga uburyo bugoye bwo gusubiza mubipimo biri hasi ugereranije nibisabwa kugirango habeho alufa-adrenergique.Harimo, anti-diuresis, ishusho rusange yibyishimo hagati harimo kuzamuka k'umuvuduko wamaraso hamwe n umuvuduko wumutima, kongera moteri, guhagarika umutima, kurakara no guhinda umushyitsi.Kubira ibyuya, isesemi no kuruka biramenyerewe nyuma yubuyobozi bwababyeyi.Na none, kuzunguruka, kubabara umutwe kuruhu byavuzwe iyo ukoresheje umunwa.

3. Mubisanzwe, uyu muti ntusabwa gukoreshwa kubagore kandi rwose ntugomba gukoreshwa mugihe utwite.Nta nubwo uyu muti usabwa gukoreshwa mu barwayi b'abana, abakuze cyangwa umutima-w'impyiko bafite amateka y'ibisebe byo mu gifu cyangwa mu nda.Ntanubwo igomba gukoreshwa ifatanije nibihindura imiti nka antidepressants, cyangwa kubarwayi bo mumutwe muri rusange.

Ibindi bicuruzwa bisa

Kongera Imibonano mpuzabitsina

Cialis (Tadalafil)
Viagra (Sildenafil)
vardenafil (Levitra)

Acetildenafil (Hongdenafil)
Yohimbine Hcl
Dapoxetine

Porogaramu

1).Imikorere mibi yimibonano mpuzabitsina -------- NIH ivuga ko hydrohloride yohimbine ari uburyo busanzwe bwa yohimbine iboneka nkumuti wandikirwa muri Amerika, kandi ko byagaragaye mubushakashatsi bwabantu kugirango bigire akamaro mukuvura imikorere mibi yumugabo.Yohimbine yerekanwe ko ifite akamaro mukuvura imikorere mibi yabagabo.Yohimbine yakoreshejwe kandi mu kuvura indwara ziterwa no guhuza ibitsina (munsi ya libido ikora) ku bagore.

2).Gutakaza ibinure -------- Yohimbine yerekanye kongera lipolysis mubushakashatsi bwinshi.Yayobowe mbere yimyitozo ngororamubiri, izamura lipolysis na serumu FFA haba mugihe cyimyitozo ikurikira;kuzibira adipocyte alpha-2 adrenoreceptors itanga byibura umusanzu uciriritse muriki gikorwa cya lipolytike.Imiyoborere mbere yo gukora imyitozo yohimbine ifite ubushobozi bwo kugabanya ibikorwa bya lipoprotein lipase yibikorwa bya adipocytes ya visceral, kongera lipolysis mububiko bwamavuta ya ginoid, no kunoza uburyo bwa lipolitike bwangiza imyitozo kubasaza.


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